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Ipamorelin vs Tesamorelin

A side-by-side research comparison of Ipamorelin and Tesamorelin across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeIpamorelinTesamorelin
Full nameIpamorelin (Selective GH Secretagogue)Tesamorelin Acetate (Egrifta)
CategoryGrowth HormoneGrowth Hormone
StatusResearch compoundFDA Approved
MechanismSelectively activates GHSR on pituitary somatotrophs. Unlike GHRP-6 and hexarelin, does not significantly activate ACTH or prolactin-releasing pathways.Binds pituitary GHRH receptors with enhanced affinity via hexenoic acid modification. Effective at mobilizing visceral fat via GH-mediated lipolysis.
Molecular weight711.9 Da5,136 Da
Half-life2 hours26-38 minutes
BioavailabilityHigh (SubQ)High (SubQ)
Typical dose100-300 mcg2 mg
Frequency1-3x dailyOnce daily
RouteSubcutaneous injectionSubcutaneous injection

Ipamorelin reported benefits

  • Clean GH release
  • No cortisol or prolactin increase
  • Improved sleep
  • Fat loss
  • Joint support
  • Anti-aging benefits

Tesamorelin reported benefits

  • Visceral fat reduction (up to 18%)
  • FDA-approved safety
  • Improved lipid panels
  • Cognitive benefits (emerging)
  • No significant IGF-1 overshoot

Related comparisons

Research and educational reference only. Not medical advice.