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Cagrilintide vs Retatrutide

A side-by-side research comparison of Cagrilintide and Retatrutide across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeCagrilintideRetatrutide
Full nameCagrilintide (AM833)Retatrutide (Triple Agonist GIP/GLP-1/Glucagon)
CategoryWeight ManagementWeight Management
StatusInvestigational (Phase III)Phase 3 Clinical Trial
MechanismActs as a dual amylin and calcitonin receptor agonist. It engages satiety centers in the area postrema and hindbrain, reducing food intake and slowing gastric emptying through a pathway distinct from GLP-1.Triple agonism creates synergistic metabolic effects. Glucagon activation increases energy expenditure and hepatic fat oxidation while GLP-1/GIP reduce appetite and improve insulin sensitivity.
Molecular weight~3963 Da5,200 Da (approximate)
Half-life~7-8 days6 days
BioavailabilityHigh via subcutaneous injectionHigh (SubQ)
Typical dose0.3-2.4 mg (titrated)1-2 mg → titrate up to 12 mg
FrequencyOnce weeklyOnce weekly
RouteSubcutaneous injectionSubcutaneous injection

Cagrilintide reported benefits

  • Appetite suppression and increased satiety
  • Meaningful weight loss
  • Complements GLP-1 agonists (additive effect)
  • Slows gastric emptying

Retatrutide reported benefits

  • Unprecedented weight loss (~24%)
  • Significant liver fat reduction
  • Improved cardiovascular markers
  • Enhanced energy expenditure
  • Superior glycemic control

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Research and educational reference only. Not medical advice.