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Cagrilintide vs Tesofensine

A side-by-side research comparison of Cagrilintide and Tesofensine across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeCagrilintideTesofensine
Full nameCagrilintide (AM833)Tesofensine (Triple Monoamine Reuptake Inhibitor)
CategoryWeight ManagementWeight Management
StatusInvestigational (Phase III)Phase 3 Clinical Trial
MechanismActs as a dual amylin and calcitonin receptor agonist. It engages satiety centers in the area postrema and hindbrain, reducing food intake and slowing gastric emptying through a pathway distinct from GLP-1.Blocks presynaptic reuptake of noradrenaline, dopamine, and serotonin in the hypothalamus, enhancing satiety signaling, reducing food reward, and increasing thermogenesis.
Molecular weight~3963 Da329.4 Da
Half-life~7-8 days8-10 days
BioavailabilityHigh via subcutaneous injectionHigh (oral ~93%)
Typical dose0.3-2.4 mg (titrated)0.25-0.5 mg
FrequencyOnce weeklyOnce daily
RouteSubcutaneous injectionOral

Cagrilintide reported benefits

  • Appetite suppression and increased satiety
  • Meaningful weight loss
  • Complements GLP-1 agonists (additive effect)
  • Slows gastric emptying

Tesofensine reported benefits

  • Significant appetite reduction
  • Increased metabolic rate
  • Improved satiety signaling
  • 10-12% body weight loss
  • Oral administration convenience

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Research and educational reference only. Not medical advice.