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MK-677 (Ibutamoren) vs Tesamorelin

A side-by-side research comparison of MK-677 (Ibutamoren) and Tesamorelin across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeMK-677 (Ibutamoren)Tesamorelin
Full nameIbutamoren Mesylate (MK-677)Tesamorelin Acetate (Egrifta)
CategoryGrowth HormoneGrowth Hormone
StatusInvestigationalFDA Approved
MechanismActs as ghrelin mimetic at GHS-R1a receptors in hypothalamus and pituitary. Excellent oral bioavailability and 24-hour duration.Binds pituitary GHRH receptors with enhanced affinity via hexenoic acid modification. Effective at mobilizing visceral fat via GH-mediated lipolysis.
Molecular weight528.7 Da5,136 Da
Half-life24 hours26-38 minutes
BioavailabilityHigh (oral)High (SubQ)
Typical dose10-25 mg2 mg
FrequencyOnce dailyOnce daily
RouteOral (capsule/liquid)Subcutaneous injection

MK-677 (Ibutamoren) reported benefits

  • Oral administration
  • Sustained 24h GH elevation
  • Increased IGF-1
  • Improved sleep depth
  • Enhanced recovery
  • Bone density support

Tesamorelin reported benefits

  • Visceral fat reduction (up to 18%)
  • FDA-approved safety
  • Improved lipid panels
  • Cognitive benefits (emerging)
  • No significant IGF-1 overshoot

Related comparisons

Research and educational reference only. Not medical advice.