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FOXO4-DRI vs SS-31 (Elamipretide)

A side-by-side research comparison of FOXO4-DRI and SS-31 (Elamipretide) across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeFOXO4-DRISS-31 (Elamipretide)
Full nameFOXO4-D-Retro-Inverso Peptide (Senolytic)SS-31 / Elamipretide (Bendavia)
CategoryAnti-AgingAnti-Aging
StatusResearch compoundInvestigational
MechanismCompetitively disrupts FOXO4 sequestration of p53 in senescent cells, releasing p53 to trigger intrinsic apoptosis selectively in cells relying on this survival mechanism.Targets cardiolipin in inner mitochondrial membrane, stabilizes cytochrome c binding, optimizes electron transfer efficiency, and reduces mitochondrial ROS by 50%.
Molecular weight~4,500 Da640.8 Da
Half-life12-24 hours (D-amino acid stability)4-6 hours
BioavailabilityModerate (SubQ)High (SubQ)
Typical dose5-10 mg/kg (animal studies)5-40 mg
Frequency3x per week for 3 weeksDaily
RouteSubcutaneousSubcutaneous or IV

FOXO4-DRI reported benefits

  • Selective senescent cell elimination
  • Potential aging reversal
  • Improved tissue function
  • Reduced inflammatory burden
  • Hair regrowth (mice)

SS-31 (Elamipretide) reported benefits

  • Mitochondrial function optimization
  • Reduced oxidative stress
  • Cardioprotection
  • Improved exercise capacity
  • Renal protection
  • Cellular energy

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Research and educational reference only. Not medical advice.