ResearchSafe

Sermorelin vs Tesamorelin

A side-by-side research comparison of Sermorelin and Tesamorelin across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeSermorelinTesamorelin
Full nameSermorelin Acetate (GHRH 1-29)Tesamorelin Acetate (Egrifta)
CategoryGrowth HormoneGrowth Hormone
StatusPreviously FDA-approved (discontinued 2008)FDA Approved
MechanismBinds GHRH receptors on anterior pituitary via cAMP-PKA pathway. Preserves natural feedback regulation and pulsatility unlike exogenous HGH.Binds pituitary GHRH receptors with enhanced affinity via hexenoic acid modification. Effective at mobilizing visceral fat via GH-mediated lipolysis.
Molecular weight3,358 Da5,136 Da
Half-life10-20 minutes26-38 minutes
BioavailabilityModerate (SubQ)High (SubQ)
Typical dose200-300 mcg2 mg
FrequencyOnce daily before bedOnce daily
RouteSubcutaneous injectionSubcutaneous injection

Sermorelin reported benefits

  • Natural GH pulsatility preserved
  • Improved sleep quality
  • Body composition improvement
  • Skin elasticity
  • Long safety record

Tesamorelin reported benefits

  • Visceral fat reduction (up to 18%)
  • FDA-approved safety
  • Improved lipid panels
  • Cognitive benefits (emerging)
  • No significant IGF-1 overshoot

Related comparisons

Research and educational reference only. Not medical advice.